WO2026038121 - USES OF A CDK2 INHIBITOR IN THE TREATMENT OF CANCER

National phase entry is expected:
Publication Number WO/2026/038121
Publication Date 19.02.2026
International Application No. PCT/IB2025/058143
International Filing Date 11.08.2025
Title **
[English] USES OF A CDK2 INHIBITOR IN THE TREATMENT OF CANCER
[French] UTILISATIONS D'UN INHIBITEUR DE CDK2 DANS LE TRAITEMENT DU CANCER
Applicants **
NOVARTIS AG
Inventors
HO, Samuel Kin Sang
MAERTENS, Ophélia
OTERO, Javier Alberto
Priority Data
63/682,037   12.08.2024   US
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Quotation for National Phase entry

Country StagesTotal
China Filing, Examination, Granting2676
EPO Filing, Examination, Granting15456
Japan Filing, Examination, Granting2525
South Korea Filing, Examination, Granting2825
USA Filing, Examination, Granting8540
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Total: 32,022
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Abstract[English] The invention relates to a pharmaceutical combination comprising a CDK2 inhibitor in combination with a CDK4 inhibitor, as well as methods of treating cancers using said combination. The present invention also relates to the use of CDK2 inhibitor in the treatment of a CCNE1 or CCNE2 amplified cancer.[French] L'invention concerne une association pharmaceutique comprenant un inhibiteur de CDK2 en association avec un inhibiteur de CDK4, ainsi que des méthodes de traitement de cancers à l'aide de ladite association. La présente invention concerne également l'utilisation d'un inhibiteur de CDK2 dans le traitement d'un cancer avec amplification de CCNE1 ou CCNE2.