WO2024028782 - NLRP3 INFLAMMASOME INHIBITORS

National phase entry is expected:
Publication Number WO/2024/028782
Publication Date 08.02.2024
International Application No. PCT/IB2023/057819
International Filing Date 02.08.2023
Title **
[English] NLRP3 INFLAMMASOME INHIBITORS
[French] INHIBITEURS DE L'INFLAMMASOME NLRP3
Applicants **
NOVARTIS AG Lichtstrasse 35 4056 Basel, CH
Inventors
GE, Xiaobin Suzhou Novartis Technical Development Co., Ltd. 18-1 Tonglian Road Bixi subdistrict Changshu Jiangsu, CN
MATTES, Henri 958 quartier le Cadeton 83570 Monfort sur Argens, FR
SHI, Zhicong China Novartis Institutes for Biomedical Research Co., Ltd. 4218 Jinke Road, Pudong New Area Shanghai, CN
XIA, Mei China Novartis Institutes for Biomedical Research Co., Ltd. 4218 Jinke Road, Pudong New Area Shanghai, CN
YE, Ning Suzhou Novartis Technical Development Co., Ltd. 18-1 Tonglian Road Bixi subdistrict Changshu Jiangsu, CN
Priority Data
63/370,300   03.08.2022   US
PCT/CN2023/097282   30.05.2023   CN
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Quotation for National Phase entry

Country StagesTotal
China Filing1646
EPO Filing, Examination6536
Japan Filing593
South Korea Filing607
USA Filing, Examination3835
MasterCard Visa

Total: 13217

The term for entry into the National Phase has expired. This quotation is for informational purposes only

Abstract[English] are defined herein, which inhibit NOD-like receptor protein 3 (NLRP3) inflammasome activity. The invention further relates to the processes for their preparation, pharmaceutical compositions and medicaments containing them, and their use in the treatment of diseases and disorders mediated by NLRP3.[French] sont tels que définis dans la description, qui inhibent l'activité de l'inflammasome de la protéine 3 du récepteur de type NOD (NLRP3). L'invention concerne en outre les procédés pour leur préparation, des compositions pharmaceutiques et des médicaments les contenant, et leur utilisation dans le traitement de maladies et de troubles médiés par NLRP3.
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