WO2022259222 - PROCESS FOR PREPARING AN ERK INHIBITOR

National phase entry:
Publication Number WO/2022/259222
Publication Date 15.12.2022
International Application No. PCT/IB2022/055416
International Filing Date 10.06.2022
Title **
[English] PROCESS FOR PREPARING AN ERK INHIBITOR
[French] PROCÉDÉ DE PRÉPARATION D'UN INHIBITEUR D'ERK
Applicants **
OTSUKA PHARMACEUTICAL CO., LTD. 2-9 Kanda Tsukasa-Machi Chiyoda-Ku, Tokyo 101-8535, JP
Inventors
BODHURI, Prabhudas c/o Astex Pharmaceuticals, Inc. 4420 Rosewood Drive, Suite 200 Pleasanton, California 94588, US
KHATRI, Hem Raj c/o Astex Pharmaceuticals, Inc. 4420 Rosewood Drive, Suite 200 Pleasanton, California 94588, US
SCOTT, Ian c/o Astex Pharmaceuticals, Inc. 4420 Rosewood Drive, Suite 200 Pleasanton, California 94588, US
READER, Michael c/o Astex Therapeutics Limited 436 Cambridge Science Park Milton Road Cambridge, Cambridgeshire CB4 0QA, GB
LATHBURY, David Charles c/o Astex Therapeutics Limited 436 Cambridge Science Park Milton Road Cambridge, Cambridgeshire CB4 0QA, GB
DAVAR, Nipun c/o Astex Pharmaceuticals, Inc. 4420 Rosewood Drive, Suite 200 Pleasanton, California 94588, US
JOHNSON, Matthew c/o Astex Pharmaceuticals, Inc. 4420 Rosewood Drive, Suite 200 Pleasanton, California 94588, US
Priority Data
63/209,877   11.06.2021   US
63/273,326   29.10.2021   US
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Quotation for National Phase entry

Country StagesTotal
China Filing2867
EPO Filing, Examination26285
Japan Filing595
South Korea Filing607
USA Filing, Examination24110
MasterCard Visa

Total: 54464

The term for entry into the National Phase has expired. This quotation is for informational purposes only

Abstract[English] The present disclosure relates generally to methods for the preparation of Compound (I).[French] La présente divulgation concerne de manière générale des procédés de préparation du composé (I).
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