WO2024246565 - PHARMACEUTICAL COMPOSITION COMPRISING IBUPROFEN

National phase entry is expected:
Publication Number WO/2024/246565
Publication Date 05.12.2024
International Application No. PCT/GR2024/000014
International Filing Date 31.05.2024
Title **
[English] PHARMACEUTICAL COMPOSITION COMPRISING IBUPROFEN
[French] COMPOSITION PHARMACEUTIQUE COMPRENANT DE L'IBUPROFÈNE
Applicants **
TSETI, Ioulia
Inventors
TSETI, Ioulia
Priority Data
20230100444   02.06.2023   GR
20230100623   27.07.2023   GR
20230100733   13.09.2023   GR
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Quotation for National Phase entry

Country StagesTotal
China Filing, Examination, Granting2221
EPO Filing, Examination, Granting7285
Japan Filing, Examination, Granting2247
South Korea Filing, Examination, Granting2325
USA Filing, Examination, Granting4740
MasterCard Visa
Total: 18,818

The term for entry into the National Phase has expired. This quotation is for informational purposes only

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Abstract[English] The present invention refers to pharmaceutical compositions comprising ibuprofen or a pharmaceutically acceptable derivative thereof and one or more solubilizing agents in the form of A) aqueous solution for use in intravenous administration comprising ibuprofen of either the sodium or lysinate salt, paracetamol and preferably one or more cyclodextrins or B) aqueous solution for use in intravenous administration wherein the one or more solubilizing agents are one or more essential amino acids and optionally one or more cyclodextrins or C) composition for use in oral administration, which comprises paracetamol and cyclodextrin, wherein said composition is in the form of either i) effervescent tablets or effervescent granules or ii) oral suspension or syrup or oral solution or iii) soft capsules.[French] La présente invention concerne des compositions pharmaceutiques comprenant de l'ibuprofène ou un dérivé pharmaceutiquement acceptable de celui-ci et un ou plusieurs agents solubilisants sous la forme de : A) une solution aqueuse destinée à être utilisée en administration intraveineuse comprenant de l'ibuprofène du sel de sodium ou de lysinate, du paracétamol et de préférence une ou plusieurs cyclodextrines ou B) une solution aqueuse destinée à être utilisée en administration intraveineuse, le ou les agents solubilisants étant un ou plusieurs acides aminés essentiels et éventuellement une ou plusieurs cyclodextrines ou C) une composition destinée à être utilisée en administration orale, qui comprend du paracétamol et de la cyclodextrine, ladite composition étant sous la forme soit i) de comprimés effervescents ou de granulés effervescents, soit ii) de suspension orale ou de sirop ou de solution orale, soit iii) de capsules molles.