WO2024121138 - CRYSTALLINE ADIPIC ACID SALT FORM OF A CCR6 ANTAGONIST

National phase entry:
Publication Number WO/2024/121138
Publication Date 13.06.2024
International Application No. PCT/EP2023/084328
International Filing Date 05.12.2023
Title **
[English] CRYSTALLINE ADIPIC ACID SALT FORM OF A CCR6 ANTAGONIST
[French] FORME DE SEL D'ACIDE ADIPIQUE CRISTALLIN D'UN ANTAGONISTE DE CCR6
Applicants **
IDORSIA PHARMACEUTICALS LTD
Inventors
FLEISCHER, Tony
MARCHAL, Daniel
RAGER, Timo
SCHAEFER, Gabriel
ZOUGGARI, Cécilia
Priority Data
PCT/EP2022/084559   06.12.2022   EP
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Quotation for National Phase entry

Country StagesTotal
China Filing, Examination, Granting2040
EPO Filing, Examination, Granting8126
Japan Filing, Examination, Granting2155
South Korea Filing, Examination, Granting2071
USA Filing, Examination, Granting5340
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Total: 19,732

The term for entry into the National Phase has expired. This quotation is for informational purposes only

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Abstract[English] The present invention relates to a crystalline form of 2-(3-{5-[(R)-(1,3-dimethyl-azetidin-3-yl)-hydroxy-(4-isopropyl- phenyl)-methyl]-pyridin-3-yl}-[1,2,4]oxadiazol-5-yl)-propan-2-ol adipic acid salt and its use in the treatment or prevention of various diseases or disorders such as cancer or inflammatory/autoimmune diseases or disorders.[French] La présente invention concerne une forme cristalline de sel d'acide adipique de 2-(3-5-[(R)-(1,3-diméthyl-azétidin-3-yl)-hydroxy-(4-isopropyl-phényl)-méthyl]-pyridin-3-yl}-[1,2,4]oxadiazol-5-yl)-propan-2-ol et son utilisation dans le traitement ou la prévention de maladies ou de troubles divers tels que le cancer ou de maladies ou de troubles inflammatoires/auto-immuns.