WO2025173034 - HYALURONIC ACID DERIVATIVES AND THEIR THERAPEUTIC USE

National phase entry is expected:
Publication Number WO/2025/173034
Publication Date 21.08.2025
International Application No. PCT/IN2025/050206
International Filing Date 13.02.2025
Title **
[English] HYALURONIC ACID DERIVATIVES AND THEIR THERAPEUTIC USE
[French] DÉRIVÉS D'ACIDE HYALURONIQUE ET LEUR UTILISATION THÉRAPEUTIQUE
Applicants **
ZYDUS LIFESCIENCES LIMITED
Inventors
DESAI, Ranjit
MITTAL, Ravindra
PANDYA, Vrajesh
JOHARAPURKAR, Amit Arvind
PUJARA, Mehul
VORA, Bhavesh
Priority Data
202421010112   14.02.2024   IN
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Quotation for National Phase entry

Country StagesTotal
China Filing, Examination, Granting2182
EPO Filing, Examination, Granting11887
Japan Filing, Examination, Granting2178
South Korea Filing, Examination, Granting2107
USA Filing, Examination, Granting9540
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Total: 27,894
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Abstract[English] The present invention relates to hyaluronic acid derivatives of the general formula (I) to which anti-inflammatory or disease-modifying drug is attached through a biodegradable linker to treat chronic degenerative diseases such as osteoarthritis or related inflammatory disorders, their pharmaceutically acceptable salts, pharmaceutical compositions containing them, methods for their preparation, use of these compounds in medicine and the intermediates involved in their preparation.[French] La présente invention concerne des dérivés d'acide hyaluronique de formule générale (I) dans laquelle un médicament anti-inflammatoire ou modificateur de maladie est fixé par l'intermédiaire d'un lieur biodégradable pour traiter des maladies dégénératives chroniques telles que l'arthrose ou des troubles inflammatoires associés, leurs sels pharmaceutiquement acceptables, des compositions pharmaceutiques les contenant, des procédés pour leur préparation, l'utilisation de ces composés en médecine et les intermédiaires impliqués dans leur préparation.

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