WO2025202864 - ENT1 INHIBITORS IN COMBINATION WITH ONCOLYTIC VIRUSES AND THEIR USE IN THE TREATMENT OF CANCER

National phase entry is expected:
Publication Number WO/2025/202864
Publication Date 02.10.2025
International Application No. PCT/IB2025/053085
International Filing Date 24.03.2025
Title **
[English] ENT1 INHIBITORS IN COMBINATION WITH ONCOLYTIC VIRUSES AND THEIR USE IN THE TREATMENT OF CANCER
[French] INHIBITEURS D'ENT1 UTILISÉS EN COMBINAISON AVEC DES VIRUS ONCOLYTIQUES ET LEUR UTILISATION DANS LE TRAITEMENT DU CANCER
Applicants **
ITEOS BELGIUM SA
Inventors
SANDERS, Theodore J.
HOUTHUYS, Erica Joke Kateligne Heleen
Priority Data
63/569,451   25.03.2024   US
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Quotation for National Phase entry

Country StagesTotal
China Filing, Examination, Granting6425
EPO Filing, Examination, Granting149297
Japan Filing, Examination, Granting5072
South Korea Filing, Examination, Granting9794
USA Filing, Examination, Granting76040
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Total: 246,628
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Abstract[English] Disclosed herein are combinations, compositions, and kits comprising an ENT1 inhibitor and an oncolytic virus. In some embodiments, the ENT1 inhibitor is a compound of Formula (I) or a pharmaceutically acceptable salt, hydrate, or solvate thereof. Also disclosed herein are methods comprising administering an ENT1 inhibitor and an oncolytic virus as well as uses of an ENT1 inhibitor and an oncolytic virus in the manufacture of a medicament. (I)[French] L'invention concerne des combinaisons, des compositions et des kits comprenant un inhibiteur d'ENT1 et un virus oncolytique. Dans certains modes de réalisation, l'inhibiteur d'ENT1 est un composé de formule (I) ou un sel, hydrate ou solvate pharmaceutiquement acceptable de celui-ci. L'invention concerne également des méthodes comprenant l'administration d'un inhibiteur d'ENT1 et d'un virus oncolytique ainsi que des utilisations d'un inhibiteur d'ENT1 et d'un virus oncolytique dans la fabrication d'un médicament. (I)

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