WO2026108953 - CARBAMATE FUMARATE, CRYSTALLINE FORM AND AMORPHOUS FORM THEREOF, AND PREPARATION METHOD THEREFOR

National phase entry is expected:
Publication Number WO/2026/108953
Publication Date 28.05.2026
International Application No. PCT/CN2025/136629
International Filing Date 21.11.2025
Title **
[English] CARBAMATE FUMARATE, CRYSTALLINE FORM AND AMORPHOUS FORM THEREOF, AND PREPARATION METHOD THEREFOR
[French] FUMARATE DE CARBAMATE, FORME CRISTALLINE ET FORME AMORPHE DE CELUI-CI, ET PROCÉDÉ DE PRÉPARATION ASSOCIÉ
[Chinese] 一种氨基甲酸酯富马酸盐及其晶型、无定型和制备方法
Applicants **
CHENGDU SHIBEIKANG BIOMEDICAL TECHNOLOGY CO., LTD.
Inventors
WANG, Xiaoyu
JIANG, Jie
FU, Haixia
MOU, Xia
TAN, Shaojun
Priority Data
202411684869.2   22.11.2024   CN
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Quotation for National Phase entry

Country StagesTotal
China Filing, Examination, Granting1692
EPO Filing, Examination, Granting11653
Japan Filing, Examination, Granting2144
South Korea Filing, Examination, Granting2050
USA Filing, Examination, Granting4740
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Total: 22,279
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Abstract[English] Provided are novel carbamate fumarate, a crystalline form and amorphous form thereof, and a preparation method therefor. The carbamate fumarate and the crystalline form and amorphous form thereof have high stability and high solubility, low hygroscopicity, and improved pharmaceutical properties, and achieves a better anti-platelet aggregation effect and higher efficacy, thereby facilitating the clinical application of drugs.[French] L'invention concerne un nouveau fumarate de carbamate, une forme cristalline et une forme amorphe de celui-ci, ainsi qu'un procédé de préparation. Le fumarate de carbamate et sa forme cristalline et sa forme amorphe ont une stabilité élevée et une solubilité élevée, une faible hygroscopicité et des propriétés pharmaceutiques améliorées, et permet d'obtenir un meilleur effet d'agrégation antiplaquettaire et une efficacité supérieure, ce qui facilite l'application clinique de médicaments.[Chinese] 提供一种新颖的氨基甲酸酯的富马酸盐,及其晶型、无定型和制备方法。所述氨基甲酸酯富马酸盐及其晶型和无定型具备较高的稳定性和溶解度、较低的引湿性,可药用性能得到提升,并且抗血小板聚集效果更好,药效更高,有利于实现药物的临床应用。

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